Assay Detail
Binding
CHEMBL4199504
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of TXK (unknown origin) using fluorescently labeled peptide as substrate after 3 hrs by microfluidic mobility shift assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Covalent Inhibitors of the TEC Family of Kinases and Their Methods of Use.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 9.53 | 9.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4206765 | — | — | 1 | 9.85 |
| CHEMBL4214683 | — | — | 1 | 9.85 |
| CHEMBL4217959 | — | — | 1 | 9.80 |
| CHEMBL4219011 | — | — | 1 | 9.74 |
| CHEMBL4203077 | — | — | 1 | 9.74 |
| CHEMBL4207292 | — | — | 1 | 9.70 |
| CHEMBL4211372 | — | — | 1 | 9.68 |
| CHEMBL4208358 | — | — | 1 | 9.66 |
| CHEMBL4216187 | — | — | 1 | 9.60 |
| CHEMBL4204572 | — | — | 1 | 9.54 |
| CHEMBL4216529 | — | — | 1 | 9.49 |
| CHEMBL4202941 | — | — | 1 | 9.41 |
| CHEMBL4215147 | — | — | 1 | 9.38 |
| CHEMBL4210857 | — | — | 1 | 9.33 |
| CHEMBL4206487 | — | — | 1 | 9.26 |
| CHEMBL4215807 | — | — | 1 | 9.23 |
| CHEMBL4218914 | — | — | 1 | 9.17 |
| CHEMBL4202618 | — | — | 1 | 9.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4206765 | — | IC50 | = | 0.14 | nM | 9.85 |
| CHEMBL4214683 | — | IC50 | = | 0.14 | nM | 9.85 |
| CHEMBL4217959 | — | IC50 | = | 0.16 | nM | 9.80 |
| CHEMBL4219011 | — | IC50 | = | 0.18 | nM | 9.74 |
| CHEMBL4203077 | — | IC50 | = | 0.18 | nM | 9.74 |
| CHEMBL4207292 | — | IC50 | = | 0.2 | nM | 9.70 |
| CHEMBL4211372 | — | IC50 | = | 0.21 | nM | 9.68 |
| CHEMBL4208358 | — | IC50 | = | 0.22 | nM | 9.66 |
| CHEMBL4216187 | — | IC50 | = | 0.25 | nM | 9.60 |
| CHEMBL4204572 | — | IC50 | = | 0.29 | nM | 9.54 |
| CHEMBL4216529 | — | IC50 | = | 0.32 | nM | 9.49 |
| CHEMBL4202941 | — | IC50 | = | 0.39 | nM | 9.41 |
| CHEMBL4215147 | — | IC50 | = | 0.42 | nM | 9.38 |
| CHEMBL4210857 | — | IC50 | = | 0.47 | nM | 9.33 |
| CHEMBL4206487 | — | IC50 | = | 0.55 | nM | 9.26 |
| CHEMBL4215807 | — | IC50 | = | 0.59 | nM | 9.23 |
| CHEMBL4218914 | — | IC50 | = | 0.67 | nM | 9.17 |
| CHEMBL4202618 | — | IC50 | = | 0.76 | nM | 9.12 |