Assay Detail
Binding
CHEMBL4232575
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant human CA9 expressed in Escherichia coli assessed as reduction in CO2 hydration by stopped flow assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis, structure and bioactivity of primary sulfamate-containing natural products.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.18 | 6.84 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3250749 | — | — | 1 | 6.84 |
| CHEMBL471144 | — | — | 1 | 5.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3250749 | — | Ki | = | 143.0 | nM | 6.84 |
| CHEMBL471144 | — | Ki | = | 3100.0 | nM | 5.51 |