Assay Detail
Functional
CHEMBL4234923
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Vasorelaxant activity in Wistar rat endothelium-denuded 3rd-order mesenteric artery assessed as reduction in norepinephrine-induced vessel contraction by myographic method
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Tissue | Artery |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Terpenoids with vasorelaxant effects from the Chinese liverwort Scapania carinthiaca.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| %max | 1 | - | - |
| EC50 | 1 | 4.43 | 4.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4246908 | — | — | 2 | 4.43 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4246908 | — | EC50 | = | 37000.0 | nM | 4.43 |
| CHEMBL4246908 | — | %max | = | 20.0 | % | - |