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Assay Detail

CHEMBL4235454

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Functional
Antiviral activity against Influenza virus assessed as inhibition of viral transcription
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism unidentified influenza virus
Confidence 1 — Organism
Curated By Intermediate

Target

unidentified influenza virus (CHEMBL613128)
Type ORGANISM
Organism unidentified influenza virus

Publication

Identification of influenza PA-Nter endonuclease inhibitors using pharmacophore- and docking-based virtual screening.
Ferro S, Gitto R, Buemi MR, Karamanou S, Stevaert A, Naesens L, De Luca L.
Bioorg Med Chem (2018) 26 : 4544 -4550
PubMed 30082105 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.37 6.37

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL463590 1 6.37

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL463590 IC50 = 430.0 nM 6.37