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Assay Detail

CHEMBL4256372

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human MCF7 cells after 24 hrs by annexin-V-FITC/propidium iodide staining based flow cytometric method
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Intermediate

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

New Hybrids Derived from Podophyllic Aldehyde and Diterpenylhydroquinones with Selectivity toward Osteosarcoma Cells.
Hernández ÁP, Díez P, García PA, Miguel Del Corral JM, Pérez-Andrés M, Díez D, San Feliciano A, Fuentes M, Castro MÁ.
ACS Med Chem Lett (2018) 9 : 328 -333
PubMed 29670695 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 4.52 4.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL23741 1 4.52
CHEMBL4282812 1 -
CHEMBL61 PODOFILOX 4.0 1 -
CHEMBL309880 PODOPHYLLIC ALDEHYDE 1 -
CHEMBL4279359 1 -
CHEMBL4284818 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL23741 IC50 = 29900.0 nM 4.52
CHEMBL4282812 IC50 > 100000.0 nM -
CHEMBL61 PODOFILOX IC50 > 100000.0 nM -
CHEMBL309880 PODOPHYLLIC ALDEHYDE IC50 > 100000.0 nM -
CHEMBL4279359 IC50 > 100000.0 nM -
CHEMBL4284818 IC50 > 100000.0 nM -