Assay Detail
Functional
CHEMBL4257029
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human NCI-H157 cells expressing mutant KRAS incubated for 72 hrs by MTS assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H157 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Compounds, compositions and methods for inhibiting cnksr1
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 5.12 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4285086 | — | — | 1 | 7.00 |
| CHEMBL4288751 | — | — | 1 | 6.30 |
| CHEMBL4278147 | — | — | 1 | 5.92 |
| CHEMBL4278841 | — | — | 1 | 5.82 |
| CHEMBL4278527 | — | — | 1 | 5.39 |
| CHEMBL4277811 | — | — | 1 | 5.28 |
| CHEMBL4277129 | — | — | 1 | 5.19 |
| CHEMBL4293956 | — | — | 1 | 5.08 |
| CHEMBL4280622 | — | — | 1 | 5.00 |
| CHEMBL4294863 | — | — | 1 | 4.83 |
| CHEMBL4293825 | — | — | 1 | 4.78 |
| CHEMBL4282291 | — | — | 1 | 4.60 |
| CHEMBL4286687 | — | — | 1 | 4.41 |
| CHEMBL4282649 | — | — | 1 | 4.26 |
| CHEMBL4283706 | — | — | 1 | 4.07 |
| CHEMBL4287729 | — | — | 1 | 4.00 |
| CHEMBL4290768 | — | — | 1 | - |
| CHEMBL4291817 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4285086 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4288751 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL4278147 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL4278841 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL4278527 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL4277811 | — | IC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL4277129 | — | IC50 | = | 6500.0 | nM | 5.19 |
| CHEMBL4293956 | — | IC50 | = | 8400.0 | nM | 5.08 |
| CHEMBL4280622 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL4294863 | — | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL4293825 | — | IC50 | = | 16600.0 | nM | 4.78 |
| CHEMBL4282291 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL4286687 | — | IC50 | = | 39100.0 | nM | 4.41 |
| CHEMBL4282649 | — | IC50 | = | 55100.0 | nM | 4.26 |
| CHEMBL4283706 | — | IC50 | = | 85000.0 | nM | 4.07 |
| CHEMBL4287729 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL4290768 | — | IC50 | - | — | - | |
| CHEMBL4291817 | — | IC50 | - | — | - |