Assay Detail
Functional
CHEMBL4257030
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human HCC515 cells expressing mutant KRAS incubated for 72 hrs by MTS assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HCC515 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Compounds, compositions and methods for inhibiting cnksr1
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 5.12 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4285086 | — | — | 1 | 7.00 |
| CHEMBL4288751 | — | — | 1 | 6.30 |
| CHEMBL4278147 | — | — | 1 | 5.92 |
| CHEMBL4278841 | — | — | 1 | 5.82 |
| CHEMBL4278527 | — | — | 1 | 5.39 |
| CHEMBL4277811 | — | — | 1 | 5.28 |
| CHEMBL4277129 | — | — | 1 | 5.19 |
| CHEMBL4293956 | — | — | 1 | 5.08 |
| CHEMBL4280622 | — | — | 1 | 5.00 |
| CHEMBL4294863 | — | — | 1 | 4.83 |
| CHEMBL4293825 | — | — | 1 | 4.78 |
| CHEMBL4282291 | — | — | 1 | 4.60 |
| CHEMBL4286687 | — | — | 1 | 4.41 |
| CHEMBL4282649 | — | — | 1 | 4.26 |
| CHEMBL4283706 | — | — | 1 | 4.07 |
| CHEMBL4287729 | — | — | 1 | 4.00 |
| CHEMBL4290768 | — | — | 1 | - |
| CHEMBL4291817 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4285086 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4288751 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL4278147 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL4278841 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL4278527 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL4277811 | — | IC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL4277129 | — | IC50 | = | 6500.0 | nM | 5.19 |
| CHEMBL4293956 | — | IC50 | = | 8400.0 | nM | 5.08 |
| CHEMBL4280622 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL4294863 | — | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL4293825 | — | IC50 | = | 16600.0 | nM | 4.78 |
| CHEMBL4282291 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL4286687 | — | IC50 | = | 39100.0 | nM | 4.41 |
| CHEMBL4282649 | — | IC50 | = | 55100.0 | nM | 4.26 |
| CHEMBL4283706 | — | IC50 | = | 85000.0 | nM | 4.07 |
| CHEMBL4287729 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL4290768 | — | IC50 | - | — | - | |
| CHEMBL4291817 | — | IC50 | - | — | - |