Assay Detail
Functional
CHEMBL4271289
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of RAS-transformed human A549 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | A549 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
From bench (laboratory) to bed (hospital/home): How to explore effective natural and synthetic PAK1-blockers/longevity-promoters for cancer therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.00 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL299496 | — | — | 1 | 6.00 |
| CHEMBL4293583 | — | — | 1 | 6.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL299496 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL4293583 | — | IC50 | = | 1000.0 | nM | 6.00 |