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Assay Detail

CHEMBL4271589

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Binding
Inhibition of ADP-BODIPY binding to Thermotoga maritima HK853 after day 1 by fluorescence polarization assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Thermotoga maritima
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Screening serine/threonine and tyrosine kinase inhibitors for histidine kinase inhibition.
Wilke KE, Fihn CA, Carlson EE.
Bioorg Med Chem (2018) 26 : 5322 -5326
PubMed 29706527 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.57 5.57

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL143307 1 5.57

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL143307 IC50 = 2700.0 nM 5.57