Assay Detail
Binding
CHEMBL4272397
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of collagen prolyl 4-hydroxylase (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Collagen Prolyl 4-Hydroxylase as a Therapeutic Target.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.74 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL167301 | — | — | 1 | 6.00 |
| CHEMBL166568 | — | — | 1 | 5.96 |
| CHEMBL88972 | PYRIDINE-2,5-DICARBOXYLIC ACID | — | 1 | 5.26 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL167301 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL166568 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL88972 | PYRIDINE-2,5-DICARBOXYLIC ACID | IC50 | = | 5500.0 | nM | 5.26 |