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Assay Detail

CHEMBL4275664

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Functional
Antiproliferative activity against human MCF7 cells assessed as reduction in cell growth after 72 hrs by sulforhodamine B assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Intermediate

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

5'-Chloro-2,2'-dihydroxychalcone and related flavanoids as treatments for prostate cancer.
Saito Y, Mizokami A, Tsurimoto H, Izumi K, Goto M, Nakagawa-Goto K.
Eur J Med Chem (2018) 157 : 1143 -1152
PubMed 30189396 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.03 5.31

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2297673 1 5.31
CHEMBL428647 PACLITAXEL 4.0 1 4.94
CHEMBL4283232 1 4.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2297673 IC50 = 4900.0 nM 5.31
CHEMBL428647 PACLITAXEL IC50 = 11500.0 nM 4.94
CHEMBL4283232 IC50 = 14100.0 nM 4.85