Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4275666

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human KBVIN cells assessed as reduction in cell growth after 72 hrs by sulforhodamine B assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

5'-Chloro-2,2'-dihydroxychalcone and related flavanoids as treatments for prostate cancer.
Saito Y, Mizokami A, Tsurimoto H, Izumi K, Goto M, Nakagawa-Goto K.
Eur J Med Chem (2018) 157 : 1143 -1152
PubMed 30189396 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.14 5.31

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2297673 1 5.31
CHEMBL4283232 1 4.96
CHEMBL428647 PACLITAXEL 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2297673 IC50 = 4900.0 nM 5.31
CHEMBL4283232 IC50 = 11100.0 nM 4.96
CHEMBL428647 PACLITAXEL IC50 = 1727400.0 nM -