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Assay Detail

CHEMBL4310788

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Anti-parasitic activity against Trypanosoma brucei gambiense MBA
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Trypanosoma brucei gambiense
Confidence 1 — Organism
Curated By Autocuration

Target

Trypanosoma brucei gambiense (CHEMBL613768)
Type ORGANISM
Organism Trypanosoma brucei gambiense

Publication

Thiazole, thio and semicarbazone derivatives against tropical infective diseases: Chagas disease, human African trypanosomiasis (HAT), leishmaniasis, and malaria.
Scarim CB, Jornada DH, Machado MGM, Ferreira CMR, Dos Santos JL, Chung MC.
Eur J Med Chem (2019) 162 : 378 -395
PubMed 30453246 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.21 7.21

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL45152 1 7.21

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL45152 IC50 = 61.0 nM 7.21