Assay Detail
ADMET
CHEMBL4312830
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Cytotoxicity against mouse 3T3L1 cells measured after 72 hrs by celltiter-glo luminescent cell viability assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Cell Type | 3T3-L1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Mechanistic Insight on the Mode of Action of Colletoic Acid.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 20 | 4.63 | 4.63 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL495841 | — | — | 1 | 4.63 |
| CHEMBL4457718 | — | — | 1 | - |
| CHEMBL4475775 | — | — | 1 | - |
| CHEMBL4566781 | — | — | 1 | - |
| CHEMBL4545661 | — | — | 1 | - |
| CHEMBL4580823 | — | — | 1 | - |
| CHEMBL4450320 | — | — | 1 | - |
| CHEMBL4436767 | — | — | 1 | - |
| CHEMBL4450502 | — | — | 1 | - |
| CHEMBL4536375 | — | — | 1 | - |
| CHEMBL4448701 | — | — | 1 | - |
| CHEMBL4528896 | — | — | 1 | - |
| CHEMBL4588470 | — | — | 1 | - |
| CHEMBL4441254 | — | — | 1 | - |
| CHEMBL4571180 | — | — | 1 | - |
| CHEMBL4529787 | — | — | 1 | - |
| CHEMBL4548901 | — | — | 1 | - |
| CHEMBL499915 | CARBENOXOLONE | 2.0 | 1 | - |
| CHEMBL4531837 | — | — | 1 | - |
| CHEMBL4552570 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL495841 | — | EC50 | = | 23550.0 | nM | 4.63 |
| CHEMBL4457718 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4475775 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4566781 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4545661 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4580823 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4450320 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4436767 | — | EC50 | > | 300000.0 | nM | - |
| CHEMBL4450502 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4536375 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4448701 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4528896 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4588470 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4441254 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4571180 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4529787 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4548901 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL499915 | CARBENOXOLONE | EC50 | > | 500000.0 | nM | - |
| CHEMBL4531837 | — | EC50 | > | 500000.0 | nM | - |
| CHEMBL4552570 | — | EC50 | > | 500000.0 | nM | - |