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Assay Detail

CHEMBL4316693

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Functional
Cytotoxicity against human SKOV3 cells
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type SK-OV-3
Confidence 1 — Organism
Curated By Autocuration

Target

SK-OV-3 (CHEMBL614925)
Type CELL-LINE
Organism Homo sapiens

Publication

Nitro-Group-Containing Drugs.
Nepali K, Lee HY, Liou JP.
J Med Chem (2019) 62 : 2851 -2893
PubMed 30295477 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 10 6.02 6.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL570892 1 6.77
CHEMBL585336 1 6.68
CHEMBL571111 1 6.36
CHEMBL568792 1 6.30
CHEMBL144896 1 5.96
CHEMBL1256927 1 5.75
CHEMBL1256965 1 5.75
CHEMBL2158186 1 5.68
CHEMBL1256966 1 5.51
CHEMBL1256989 1 5.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL570892 IC50 = 170.0 nM 6.77
CHEMBL585336 IC50 = 210.0 nM 6.68
CHEMBL571111 IC50 = 440.0 nM 6.36
CHEMBL568792 IC50 = 500.0 nM 6.30
CHEMBL144896 IC50 = 1100.0 nM 5.96
CHEMBL1256927 IC50 = 1800.0 nM 5.75
CHEMBL1256965 IC50 = 1800.0 nM 5.75
CHEMBL2158186 IC50 = 2100.0 nM 5.68
CHEMBL1256966 IC50 = 3100.0 nM 5.51
CHEMBL1256989 IC50 = 3300.0 nM 5.48