Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4317089

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human MCF7 cells after 72 hrs by SRB assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Autocuration

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis of new derivatives of boehmeriasin A and their biological evaluation in liver cancer.
Güzelcan EA, Baxendale IR, Cetin-Atalay R, Baumann M.
Eur J Med Chem (2019) 166 : 243 -255
PubMed 30716712 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 7.59 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4446479 1 9.00
CHEMBL1958071 1 8.30
CHEMBL4439007 1 7.80
CHEMBL1958076 1 7.68
CHEMBL4443083 1 5.16
CHEMBL4438041 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4446479 IC50 = 1.0 nM 9.00
CHEMBL1958071 IC50 = 5.0 nM 8.30
CHEMBL4439007 IC50 = 16.0 nM 7.80
CHEMBL1958076 IC50 = 21.0 nM 7.68
CHEMBL4443083 IC50 = 7000.0 nM 5.16
CHEMBL4438041 IC50 - -