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Assay Detail

CHEMBL4317094

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human FOCUS cells after 72 hrs by SRB assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Synthesis of new derivatives of boehmeriasin A and their biological evaluation in liver cancer.
Güzelcan EA, Baxendale IR, Cetin-Atalay R, Baumann M.
Eur J Med Chem (2019) 166 : 243 -255
PubMed 30716712 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.97 7.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4446479 1 7.92
CHEMBL1958071 1 7.70
CHEMBL4443083 1 5.30
CHEMBL4438041 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4446479 IC50 = 12.0 nM 7.92
CHEMBL1958071 IC50 = 20.0 nM 7.70
CHEMBL4443083 IC50 = 5000.0 nM 5.30
CHEMBL4438041 IC50 - -