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Assay Detail

CHEMBL4317096

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human MCF10A cells after 72 hrs by SRB assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type MCF-10A
Confidence 1 — Organism
Curated By Autocuration

Target

MCF-10A (CHEMBL614321)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis of new derivatives of boehmeriasin A and their biological evaluation in liver cancer.
Güzelcan EA, Baxendale IR, Cetin-Atalay R, Baumann M.
Eur J Med Chem (2019) 166 : 243 -255
PubMed 30716712 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 6.63 6.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1958071 1 6.85
CHEMBL1958076 1 6.85
CHEMBL4446479 1 6.70
CHEMBL4439007 1 6.10
CHEMBL4438041 1 -
CHEMBL4443083 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1958071 IC50 = 140.0 nM 6.85
CHEMBL1958076 IC50 = 140.0 nM 6.85
CHEMBL4446479 IC50 = 200.0 nM 6.70
CHEMBL4439007 IC50 = 800.0 nM 6.10
CHEMBL4438041 IC50 - -
CHEMBL4443083 IC50 - -