Assay Detail
Binding
CHEMBL4322155
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human TASK1 expressed in CHO cells by Inside-out macro-patches based electrophysiology assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Potassium channel subfamily K member 3 (CHEMBL2321613) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
TASK Channels Pharmacology: New Challenges in Drug Design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.15 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL148342 | — | — | 1 | 8.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL148342 | — | IC50 | = | 7.0 | nM | 8.15 |