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Assay Detail

CHEMBL4324435

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to AhR (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Aryl hydrocarbon receptor (CHEMBL3201)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Targeting Aryl hydrocarbon receptor for next-generation immunotherapies: Selective modulators (SAhRMs) versus rapidly metabolized ligands (RMAhRLs).
Dolciami D, Ballarotto M, Gargaro M, López-Cara LC, Fallarino F, Macchiarulo A.
Eur J Med Chem (2020) 185 : 111842 -111842
PubMed 31727470 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 9.89 9.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4580482 1 9.89

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4580482 Kd = 0.13 nM 9.89