Assay Detail
Functional
CHEMBL4325428
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Antiproliferative activity against human MV4-11 cells measured after 3 days by celltiter-glo luminescence assay
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MV4-11 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of Highly Potent, Selective, and Orally Efficacious p300/CBP Histone Acetyltransferases Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 28 | 7.64 | 8.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4457144 | — | — | 1 | 8.54 |
| CHEMBL4567310 | — | — | 1 | 8.46 |
| CHEMBL4474109 | — | — | 1 | 8.43 |
| CHEMBL4475351 | — | — | 1 | 8.40 |
| CHEMBL4587968 | — | — | 1 | 8.38 |
| CHEMBL4449940 | — | — | 1 | 8.32 |
| CHEMBL4449592 | — | — | 1 | 8.09 |
| CHEMBL4552724 | — | — | 1 | 8.06 |
| CHEMBL4593536 | — | — | 1 | 7.97 |
| CHEMBL4474031 | — | — | 1 | 7.92 |
| CHEMBL4450724 | — | — | 1 | 7.87 |
| CHEMBL4439084 | — | — | 1 | 7.80 |
| CHEMBL4452911 | — | — | 1 | 7.69 |
| CHEMBL4464962 | — | — | 1 | 7.60 |
| CHEMBL4524352 | — | — | 1 | 7.19 |
| CHEMBL4584269 | — | — | 1 | 7.14 |
| CHEMBL4513653 | — | — | 1 | 7.11 |
| CHEMBL4456527 | — | — | 1 | 6.93 |
| CHEMBL4472048 | — | — | 1 | 6.81 |
| CHEMBL4441280 | — | — | 1 | 6.69 |
| CHEMBL4282264 | A-485 | — | 1 | 6.59 |
| CHEMBL4519167 | — | — | 1 | 6.08 |
| CHEMBL4582713 | — | — | 1 | - |
| CHEMBL4566439 | — | — | 1 | - |
| CHEMBL4436959 | — | — | 1 | - |
| CHEMBL4446240 | — | — | 1 | - |
| CHEMBL4464151 | — | — | 1 | - |
| CHEMBL4525368 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4457144 | — | IC50 | = | 2.9 | nM | 8.54 |
| CHEMBL4567310 | — | IC50 | = | 3.5 | nM | 8.46 |
| CHEMBL4474109 | — | IC50 | = | 3.7 | nM | 8.43 |
| CHEMBL4475351 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4587968 | — | IC50 | = | 4.2 | nM | 8.38 |
| CHEMBL4449940 | — | IC50 | = | 4.8 | nM | 8.32 |
| CHEMBL4449592 | — | IC50 | = | 8.2 | nM | 8.09 |
| CHEMBL4552724 | — | IC50 | = | 8.8 | nM | 8.06 |
| CHEMBL4593536 | — | IC50 | = | 10.7 | nM | 7.97 |
| CHEMBL4474031 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL4450724 | — | IC50 | = | 13.5 | nM | 7.87 |
| CHEMBL4439084 | — | IC50 | = | 15.8 | nM | 7.80 |
| CHEMBL4452911 | — | IC50 | = | 20.4 | nM | 7.69 |
| CHEMBL4464962 | — | IC50 | = | 24.9 | nM | 7.60 |
| CHEMBL4524352 | — | IC50 | = | 64.3 | nM | 7.19 |
| CHEMBL4584269 | — | IC50 | = | 72.8 | nM | 7.14 |
| CHEMBL4513653 | — | IC50 | = | 77.0 | nM | 7.11 |
| CHEMBL4456527 | — | IC50 | = | 118.0 | nM | 6.93 |
| CHEMBL4472048 | — | IC50 | = | 156.3 | nM | 6.81 |
| CHEMBL4441280 | — | IC50 | = | 206.0 | nM | 6.69 |
| CHEMBL4282264 | A-485 | IC50 | = | 255.2 | nM | 6.59 |
| CHEMBL4519167 | — | IC50 | = | 825.0 | nM | 6.08 |
| CHEMBL4582713 | — | IC50 | > | 500.0 | nM | - |
| CHEMBL4566439 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL4436959 | — | IC50 | - | — | - | |
| CHEMBL4446240 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL4464151 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL4525368 | — | IC50 | > | 5000.0 | nM | - |