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Assay Detail

CHEMBL4333750

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antifungal activity against azole-resistant Candida albicans after 24 hrs by resazurin dye based fluorimetric assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Candida albicans
Confidence 1 — Organism
Curated By Autocuration

Target

Candida albicans (CHEMBL366)
Type ORGANISM
Organism Candida albicans

Publication

Synthesis and antimicrobial activities of N<sup>6</sup>-hydroxyagelasine analogs and revision of the structure of ageloximes.
Paulsen B, Fredriksen KA, Petersen D, Maes L, Matheeussen A, Naemi AO, Scheie AA, Simm R, Ma R, Wan B, Franzblau S, Gundersen LL.
Bioorg Med Chem (2019) 27 : 620 -629
PubMed 30638761 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.73 6.39

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1463 FLUCYTOSINE 4.0 1 6.39
CHEMBL4592498 1 5.70
CHEMBL4469221 1 5.10
CHEMBL4443174 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1463 FLUCYTOSINE IC50 = 410.0 nM 6.39
CHEMBL4592498 IC50 = 2000.0 nM 5.70
CHEMBL4469221 IC50 = 8000.0 nM 5.10
CHEMBL4443174 IC50 > 64000.0 nM -