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Assay Detail

CHEMBL4335394

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Gaussia tagged Influenza A virus (A/Puerto Rico/8/34(H1N1)) infected in MDCK cells assessed as inhibition of H1N1 replication measured at 24 hrs post infection by luciferase reporter gene assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Influenza A virus
Confidence 1 — Organism
Curated By Autocuration

Target

Influenza A virus (CHEMBL613740)
Type ORGANISM
Organism Influenza A virus

Publication

Discovery, Optimization, and Target Identification of Novel Potent Broad-Spectrum Antiviral Inhibitors.
Yang Y, Cao L, Gao H, Wu Y, Wang Y, Fang F, Lan T, Lou Z, Rao Y.
J Med Chem (2019) 62 : 4056 -4073
PubMed 30938999 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.62 6.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4454780 1 6.62

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4454780 EC50 = 240.0 nM 6.62