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Assay Detail

CHEMBL4335417

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCV infected in human Huh7.5.1 cells assessed as decrease in viral infection
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Discovery, Optimization, and Target Identification of Novel Potent Broad-Spectrum Antiviral Inhibitors.
Yang Y, Cao L, Gao H, Wu Y, Wang Y, Fang F, Lan T, Lou Z, Rao Y.
J Med Chem (2019) 62 : 4056 -4073
PubMed 30938999 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.82 7.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4454780 1 7.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4454780 EC50 = 15.0 nM 7.82