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Assay Detail

CHEMBL4335801

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Functional
Inhibition of cell migration in human HUVEC cells assessed as decrease in cell velocity measured after 16 hrs by crystal violet staining based scratch assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HUVEC
Confidence 1 — Organism
Curated By Autocuration

Target

HUVEC (CHEMBL613979)
Type CELL-LINE
Organism Homo sapiens

Publication

Chivosazole A Modulates Protein-Protein Interactions of Actin.
Wang S, Gegenfurtner FA, Crevenna AH, Ziegenhain C, Kliesmete Z, Enard W, Müller R, Vollmar AM, Schneider S, Zahler S.
J Nat Prod (2019) 82 : 1961 -1970
PubMed 31260301 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.91 7.50

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4522174 1 7.50
CHEMBL411879 LATRUNCULIN B 1 6.32

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4522174 IC50 = 31.68 nM 7.50
CHEMBL411879 LATRUNCULIN B IC50 = 478.0 nM 6.32