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Assay Detail

CHEMBL4336768

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of CK1delta/CK1epsilon (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 7 — Homologous single protein target
Curated By Autocuration

Target

Casein kinase I delta/epsilon (CHEMBL3038494)
Type PROTEIN COMPLEX
Organism Homo sapiens

Publication

Small molecule modulators targeting protein kinase CK1 and CK2.
Qiao Y, Chen T, Yang H, Chen Y, Lin H, Qu W, Feng F, Liu W, Guo Q, Liu Z, Sun H.
Eur J Med Chem (2019) 181 : 111581 -111581
PubMed 31400711 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.00 6.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL404941 1 6.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL404941 IC50 = 1000.0 nM 6.00