Assay Detail
Binding
CHEMBL4337203
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Inhibition of human MAOA
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Multi-target-directed-ligands acting as enzyme inhibitors and receptor ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.10 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1929421 | — | — | 1 | 9.52 |
| CHEMBL4173258 | — | — | 1 | 6.84 |
| CHEMBL14638 | CIPROXIFAN | — | 1 | 4.94 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1929421 | — | IC50 | = | 0.3 | nM | 9.52 |
| CHEMBL4173258 | — | IC50 | = | 145.0 | nM | 6.84 |
| CHEMBL14638 | CIPROXIFAN | IC50 | = | 11400.0 | nM | 4.94 |