Assay Detail
Binding
CHEMBL4338733
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Binding affinity to human neurotensin receptor 1
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Fluorescence Labeling of Neurotensin(8-13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 9.28 | 9.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL415788 | — | — | 1 | 9.62 |
| CHEMBL4579623 | — | — | 1 | 9.29 |
| CHEMBL407196 | NEUROTENSIN | — | 1 | 8.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL415788 | — | Ki | = | 0.24 | nM | 9.62 |
| CHEMBL4579623 | — | Ki | = | 0.51 | nM | 9.29 |
| CHEMBL407196 | NEUROTENSIN | Ki | = | 1.2 | nM | 8.92 |