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Assay Detail

CHEMBL4339112

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human N-terminal GST-tagged IDO1 expressed in Escherichia coli Rosetta(DE3) pLysS using L-tryptophan as substrate measured after 1 hr by fluorescence assay
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Indoleamine 2,3-dioxygenase 1 (CHEMBL4685)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of Hydroxyamidine Based Inhibitors of IDO1 for Cancer Immunotherapy with Reduced Potential for Glucuronidation.
Steeneck C, Kinzel O, Anderhub S, Hornberger M, Pinto S, Morschhaeuser B, Braun F, Kleymann G, Hoffmann T.
ACS Med Chem Lett (2020) 11 : 179 -187
PubMed 32071686 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 26 6.92 7.68

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4585089 1 7.68
CHEMBL4441030 1 7.52
CHEMBL4578545 1 7.21
CHEMBL4437616 1 7.16
CHEMBL4448442 1 7.15
CHEMBL3545369 EPACADOSTAT 3.0 1 7.14
CHEMBL4455438 1 7.14
CHEMBL4439896 1 7.08
CHEMBL4451194 1 7.03
CHEMBL4549976 1 7.03
CHEMBL4441246 1 7.00
CHEMBL4434929 1 6.96
CHEMBL4475499 1 6.89
CHEMBL4452336 1 6.89
CHEMBL4521926 1 6.85
CHEMBL4449948 1 6.85
CHEMBL4436560 1 6.85
CHEMBL4465837 1 6.82
CHEMBL4483087 1 6.82
CHEMBL4538516 1 6.75
CHEMBL584991 1 6.68
CHEMBL4545974 1 6.64
CHEMBL4461796 1 6.62
CHEMBL4533342 1 6.57
CHEMBL4533432 1 6.44
CHEMBL4573030 1 6.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4585089 IC50 = 21.0 nM 7.68
CHEMBL4441030 IC50 = 30.0 nM 7.52
CHEMBL4578545 IC50 = 61.0 nM 7.21
CHEMBL4437616 IC50 = 70.0 nM 7.16
CHEMBL4448442 IC50 = 71.0 nM 7.15
CHEMBL3545369 EPACADOSTAT IC50 = 73.0 nM 7.14
CHEMBL4455438 IC50 = 73.0 nM 7.14
CHEMBL4439896 IC50 = 84.0 nM 7.08
CHEMBL4451194 IC50 = 93.0 nM 7.03
CHEMBL4549976 IC50 = 93.0 nM 7.03
CHEMBL4441246 IC50 = 100.0 nM 7.00
CHEMBL4434929 IC50 = 110.0 nM 6.96
CHEMBL4475499 IC50 = 130.0 nM 6.89
CHEMBL4452336 IC50 = 130.0 nM 6.89
CHEMBL4521926 IC50 = 140.0 nM 6.85
CHEMBL4449948 IC50 = 140.0 nM 6.85
CHEMBL4436560 IC50 = 140.0 nM 6.85
CHEMBL4465837 IC50 = 150.0 nM 6.82
CHEMBL4483087 IC50 = 150.0 nM 6.82
CHEMBL4538516 IC50 = 180.0 nM 6.75
CHEMBL584991 IC50 = 210.0 nM 6.68
CHEMBL4545974 IC50 = 230.0 nM 6.64
CHEMBL4461796 IC50 = 240.0 nM 6.62
CHEMBL4533342 IC50 = 270.0 nM 6.57
CHEMBL4533432 IC50 = 360.0 nM 6.44
CHEMBL4573030 IC50 = 560.0 nM 6.25