Assay Detail
Binding
CHEMBL4345202
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to wild type human partial length PIP5K1C (M1 to T668 residues) expressed in mammalian expression system by Kinomescan method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma (CHEMBL1908383) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.58 | 6.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4452939 | — | — | 1 | 6.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4452939 | — | Kd | = | 260.0 | nM | 6.58 |