Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4346799

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of CDK9 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cyclin-dependent kinase 9 (CHEMBL3116)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Cyclin-Dependent Kinase 2 Inhibitors in Cancer Therapy: An Update.
Tadesse S, Caldon EC, Tilley W, Wang S.
J Med Chem (2019) 62 : 4233 -4251
PubMed 30543440 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.58 7.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4579344 1 7.58

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4579344 IC50 = 26.0 nM 7.58