Assay Detail
Functional
CHEMBL4347502
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Antiproliferative activity against human HT-29 cells incubated for 2 days by MTT assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HT-29 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Novel multitarget inhibitors with antiangiogenic and immunomodulator properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 5.04 | 6.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4535136 | — | — | 1 | 6.28 |
| CHEMBL4586070 | — | — | 1 | 5.82 |
| CHEMBL4439814 | — | — | 1 | 5.46 |
| CHEMBL535 | SUNITINIB | 4.0 | 1 | 5.42 |
| CHEMBL4452195 | — | — | 1 | 4.92 |
| CHEMBL4445564 | — | — | 1 | 4.85 |
| CHEMBL1336 | SORAFENIB | 4.0 | 1 | 4.77 |
| CHEMBL4099869 | — | — | 1 | 4.72 |
| CHEMBL4472839 | — | — | 1 | 4.70 |
| CHEMBL4570579 | — | — | 1 | 4.70 |
| CHEMBL4524155 | — | — | 1 | 4.48 |
| CHEMBL4448636 | — | — | 1 | 4.33 |
| CHEMBL4578275 | — | — | 1 | - |
| CHEMBL4593366 | — | — | 1 | - |
| CHEMBL4459023 | — | — | 1 | - |
| CHEMBL4529831 | — | — | 1 | - |
| CHEMBL4448455 | — | — | 1 | - |
| CHEMBL4581003 | — | — | 1 | - |
| CHEMBL4579588 | — | — | 1 | - |
| CHEMBL4590349 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4535136 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL4586070 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL4439814 | — | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL535 | SUNITINIB | IC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL4452195 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL4445564 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL4099869 | — | IC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL4472839 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL4570579 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL4524155 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL4448636 | — | IC50 | = | 47000.0 | nM | 4.33 |
| CHEMBL4578275 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4593366 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4459023 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4529831 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4448455 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4581003 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4579588 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4590349 | — | IC50 | > | 200000.0 | nM | - |