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Assay Detail

CHEMBL4348089

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Functional
Antiviral activity against HSV-1 infected in African green monkey Vero cells preincubated with virus for 5 mins
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 1
Cell Type Vero
Confidence 1 — Organism
Curated By Autocuration

Target

Human alphaherpesvirus 1 (CHEMBL377)
Type ORGANISM
Organism Human alphaherpesvirus 1

Publication

Compounds based on 5-(perylen-3-ylethynyl)uracil scaffold: High activity against tick-borne encephalitis virus and non-specific activity against enterovirus A.
Chistov AA, Orlov AA, Streshnev PP, Slesarchuk NA, Aparin IO, Rathi B, Brylev VA, Kutyakov SV, Mikhura IV, Ustinov AV, Westman G, Palyulin VA, Jain N, Osolodkin DI, Kozlovskaya LI, Korshun VA.
Eur J Med Chem (2019) 171 : 93 -103
PubMed 30909022 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 7.45 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3797928 1 8.70
CHEMBL3798024 1 7.32
CHEMBL4472240 1 7.06
CHEMBL4473048 1 6.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3797928 EC50 = 2.0 nM 8.70
CHEMBL3798024 EC50 = 48.0 nM 7.32
CHEMBL4472240 EC50 = 87.0 nM 7.06
CHEMBL4473048 EC50 = 190.0 nM 6.72