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Assay Detail

CHEMBL4348093

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Functional
Antiviral activity against VSV infected in African green monkey Vero cells assessed as plaque reduction preincubated for 10 mins inocula removed after 1 hr followed by overlaying with 2% methylcellulose and measured after 1 to 2 days by crystal violet staining based assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vesicular stomatitis virus
Cell Type Vero
Confidence 1 — Organism
Curated By Autocuration

Target

Vesicular stomatitis virus (CHEMBL613739)
Type ORGANISM
Organism Vesicular stomatitis virus

Publication

Compounds based on 5-(perylen-3-ylethynyl)uracil scaffold: High activity against tick-borne encephalitis virus and non-specific activity against enterovirus A.
Chistov AA, Orlov AA, Streshnev PP, Slesarchuk NA, Aparin IO, Rathi B, Brylev VA, Kutyakov SV, Mikhura IV, Ustinov AV, Westman G, Palyulin VA, Jain N, Osolodkin DI, Kozlovskaya LI, Korshun VA.
Eur J Med Chem (2019) 171 : 93 -103
PubMed 30909022 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 8.70 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3797928 1 8.70
CHEMBL3798024 1 8.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3797928 EC50 = 2.0 nM 8.70
CHEMBL3798024 EC50 = 2.0 nM 8.70