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Assay Detail

CHEMBL4348095

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Functional
Antiviral activity against influenza A virus H3N2 infected in dog MDCK cells assessed as plaque reduction preincubated for 10 mins inocula removed after 1 hr followed by overlaying with 0.8% agarose and measured after 1 to 2 days by crystal violet staining based assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Influenza A virus
Confidence 1 — Organism
Curated By Autocuration

Target

Influenza A virus (CHEMBL613740)
Type ORGANISM
Organism Influenza A virus

Publication

Compounds based on 5-(perylen-3-ylethynyl)uracil scaffold: High activity against tick-borne encephalitis virus and non-specific activity against enterovirus A.
Chistov AA, Orlov AA, Streshnev PP, Slesarchuk NA, Aparin IO, Rathi B, Brylev VA, Kutyakov SV, Mikhura IV, Ustinov AV, Westman G, Palyulin VA, Jain N, Osolodkin DI, Kozlovskaya LI, Korshun VA.
Eur J Med Chem (2019) 171 : 93 -103
PubMed 30909022 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 8.70 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3797928 1 8.70
CHEMBL3798024 1 8.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3797928 EC50 = 2.0 nM 8.70
CHEMBL3798024 EC50 = 2.0 nM 8.70