Assay Detail
Binding
CHEMBL4355048
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Binding affinity to HIV1 TAR RNA
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Human immunodeficiency virus 1 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthetic small-molecule RNA ligands: future prospects as therapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 5.42 | 5.87 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1572 | NETILMICIN | 4.0 | 1 | 5.87 |
| CHEMBL4474530 | — | — | 1 | 5.62 |
| CHEMBL4442026 | — | — | 1 | 4.76 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1572 | NETILMICIN | Kd | = | 1350.0 | nM | 5.87 |
| CHEMBL4474530 | — | Kd | = | 2400.0 | nM | 5.62 |
| CHEMBL4442026 | — | Kd | = | 17500.0 | nM | 4.76 |