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Assay Detail

CHEMBL4355057

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCV infected in MDCK cells assessed as reduction in viral replication
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Synthetic small-molecule RNA ligands: future prospects as therapeutic agents.
Di Giorgio A, Duca M.
Medchemcomm (2019) 10 : 1242 -1255
PubMed 31534649 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 4.15 4.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1226 AMINODIMETHOXYQUINAZOLINYLPIPERAZINE 1 4.15

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1226 AMINODIMETHOXYQUINAZOLINYLPIPERAZINE EC50 = 71000.0 nM 4.15