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Assay Detail

CHEMBL4357660

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Plasmodium falciparum HAP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Plasmodium falciparum
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Plasmepsin Inhibitors in Antimalarial Drug Discovery: Medicinal Chemistry and Target Validation (2000 to Present).
Cheuka PM, Dziwornu G, Okombo J, Chibale K.
J Med Chem (2020) 63 : 4445 -4467
PubMed 31913032 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.16 6.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4516552 1 6.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4516552 IC50 = 690.0 nM 6.16