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Assay Detail

CHEMBL4364495

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human HeLa Cells
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

HeLa (CHEMBL399)
Type CELL-LINE
Organism Homo sapiens

Publication

Developments in the anticancer activity of structurally modified curcumin: An up-to-date review.
Rodrigues FC, Anil Kumar NV, Thakur G.
Eur J Med Chem (2019) 177 : 76 -104
PubMed 31129455 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.08 5.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL53463 DOXORUBICIN 4.0 1 5.70
CHEMBL4517144 1 4.90
CHEMBL557311 1 4.85
CHEMBL140 CURCUMIN 3.0 1 4.85
CHEMBL4435732 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL53463 DOXORUBICIN IC50 = 2020.0 nM 5.70
CHEMBL4517144 IC50 = 12470.0 nM 4.90
CHEMBL557311 IC50 = 14030.0 nM 4.85
CHEMBL140 CURCUMIN IC50 = 14030.0 nM 4.85
CHEMBL4435732 IC50 > 10000.0 nM -