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Assay Detail

CHEMBL4376314

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against Plasmodium falciparum Dd2 by HRP2 assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Primaquine derivatives: Modifications of the terminal amino group.
Zorc B, Perković I, Pavić K, Rajić Z, Beus M.
Eur J Med Chem (2019) 182 : 111640 -111640
PubMed 31472472 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.11 5.11

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4522595 1 5.11
CHEMBL4460395 1 5.11
CHEMBL4463583 1 5.11
CHEMBL4593843 1 5.11
CHEMBL4449670 1 5.11
CHEMBL4445381 1 5.11

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4522595 IC50 = 7740.0 nM 5.11
CHEMBL4460395 IC50 = 7740.0 nM 5.11
CHEMBL4463583 IC50 = 7740.0 nM 5.11
CHEMBL4593843 IC50 = 7740.0 nM 5.11
CHEMBL4449670 IC50 = 7740.0 nM 5.11
CHEMBL4445381 IC50 = 7740.0 nM 5.11