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Assay Detail

CHEMBL4376915

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Functional
Antiviral activity against Respiratory syncytial virus
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Respiratory syncytial virus
Confidence 1 — Organism
Curated By Autocuration

Target

Respiratory syncytial virus (CHEMBL612679)
Type ORGANISM
Organism Respiratory syncytial virus

Publication

State of the Art in Respiratory Syncytial Virus Drug Discovery and Development.
Cockerill GS, Good JAD, Mathews N.
J Med Chem (2019) 62 : 3206 -3227
PubMed 30411898 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 9 8.32 9.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4528752 1 9.82
CHEMBL4435108 1 9.25
CHEMBL4297497 SISUNATOVIR 2.0 1 8.89
CHEMBL4458694 1 8.56
CHEMBL4542924 1 8.00
CHEMBL4469438 1 7.51
CHEMBL4540519 1 6.18
CHEMBL4522047 1 -
CHEMBL4475481 ZELICAPAVIR 2.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4528752 EC50 = 0.15 nM 9.82
CHEMBL4435108 EC50 = 0.56 nM 9.25
CHEMBL4297497 SISUNATOVIR EC50 = 1.3 nM 8.89
CHEMBL4458694 EC50 = 2.75 nM 8.56
CHEMBL4542924 EC50 = 10.0 nM 8.00
CHEMBL4469438 EC50 = 31.0 nM 7.51
CHEMBL4540519 EC50 = 660.0 nM 6.18
CHEMBL4522047 EC50 < 1000.0 nM -
CHEMBL4475481 ZELICAPAVIR EC50 < 400.0 nM -