Assay Detail
Binding
CHEMBL4380527
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Inhibition of wild-type human partial length ULK1 (M1 to T309 residues) expressed in mammalian expression system by Kinomescan method
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Serine/threonine-protein kinase ULK1 (CHEMBL6006) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of BAY-985, a Highly Selective TBK1/IKKε Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 6.49 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4435393 | — | — | 1 | 8.05 |
| CHEMBL4468020 | — | — | 1 | 7.55 |
| CHEMBL4543618 | — | — | 1 | 6.58 |
| CHEMBL4566796 | — | — | 1 | 6.43 |
| CHEMBL4454902 | — | — | 1 | 6.38 |
| CHEMBL4538751 | — | — | 1 | 6.01 |
| CHEMBL4594167 | — | — | 1 | 5.79 |
| CHEMBL4537673 | BAY-985 | — | 1 | 5.10 |
| CHEMBL4553949 | — | — | 1 | - |
| CHEMBL4466150 | — | — | 1 | - |
| CHEMBL4547610 | — | — | 1 | - |
| CHEMBL4436416 | — | — | 1 | - |
| CHEMBL4453481 | — | — | 1 | - |
| CHEMBL4436188 | — | — | 1 | - |
| CHEMBL4515413 | — | — | 1 | - |
| CHEMBL4549459 | — | — | 1 | - |
| CHEMBL4552254 | — | — | 1 | - |
| CHEMBL4453292 | — | — | 1 | - |
| CHEMBL4538591 | BAY-440 | — | 1 | - |
| CHEMBL4451595 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4435393 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL4468020 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL4543618 | — | IC50 | = | 263.0 | nM | 6.58 |
| CHEMBL4566796 | — | IC50 | = | 368.0 | nM | 6.43 |
| CHEMBL4454902 | — | IC50 | = | 416.0 | nM | 6.38 |
| CHEMBL4538751 | — | IC50 | = | 980.0 | nM | 6.01 |
| CHEMBL4594167 | — | IC50 | = | 1640.0 | nM | 5.79 |
| CHEMBL4537673 | BAY-985 | IC50 | = | 7930.0 | nM | 5.10 |
| CHEMBL4553949 | — | IC50 | - | — | - | |
| CHEMBL4466150 | — | IC50 | - | — | - | |
| CHEMBL4547610 | — | IC50 | - | — | - | |
| CHEMBL4436416 | — | IC50 | - | — | - | |
| CHEMBL4453481 | — | IC50 | - | — | - | |
| CHEMBL4436188 | — | IC50 | - | — | - | |
| CHEMBL4515413 | — | IC50 | - | — | - | |
| CHEMBL4549459 | — | IC50 | - | — | - | |
| CHEMBL4552254 | — | IC50 | - | — | - | |
| CHEMBL4453292 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4538591 | BAY-440 | IC50 | - | — | - | |
| CHEMBL4451595 | — | IC50 | - | — | - |