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Assay Detail

CHEMBL4380852

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Functional
Antiproliferative activity against human OCI-LY7 cells assessed as reduction in cell viability incubated for 72 hrs by CCK8 assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type OCI-Ly7
Confidence 1 — Organism
Curated By Autocuration

Target

OCI-Ly7 (CHEMBL4523564)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis and Biological Evaluation of B-Cell Lymphoma 6 Inhibitors of N-Phenyl-4-pyrimidinamine Derivatives Bearing Potent Activities against Tumor Growth.
Guo W, Xing Y, Zhang Q, Xie J, Huang D, Gu H, He P, Zhou M, Xu S, Pang X, Liu M, Yi Z, Chen Y.
J Med Chem (2020) 63 : 676 -695
PubMed 31895575 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.89 5.79

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4538610 1 5.79
CHEMBL4077392 1 4.47
CHEMBL4061302 1 4.41

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4538610 IC50 = 1620.0 nM 5.79
CHEMBL4077392 IC50 = 33900.0 nM 4.47
CHEMBL4061302 IC50 = 39000.0 nM 4.41