Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4385019

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human AZ-521 cells assessed as reduction in cell viability after 48 hrs by MTT assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type AZ-521
Confidence 1 — Organism
Curated By Autocuration

Target

AZ-521 cell line (CHEMBL614274)
Type CELL-LINE
Organism Homo sapiens

Publication

Melanogenesis-Inhibitory and Cytotoxic Activities of Triterpene Glycoside Constituents from the Bark of Albizia procera.
Zhang J, Akihisa T, Kurita M, Kikuchi T, Zhu WF, Ye F, Dong ZH, Liu WY, Feng F, Xu J.
J Nat Prod (2018) 81 : 2612 -2620
PubMed 30520635 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 6.12 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4451985 1 6.40
CHEMBL4483588 1 6.30
CHEMBL4581280 1 6.22
CHEMBL4448517 1 5.92
CHEMBL4561300 1 5.77

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4451985 IC50 = 400.0 nM 6.40
CHEMBL4483588 IC50 = 500.0 nM 6.30
CHEMBL4581280 IC50 = 600.0 nM 6.22
CHEMBL4448517 IC50 = 1200.0 nM 5.92
CHEMBL4561300 IC50 = 1700.0 nM 5.77