Assay Detail
Functional
CHEMBL4390734
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Growth inhibition of Microcystis aeruginosa FACHB905 incubated for 7 days
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Microcystis aeruginosa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Design, synthesis and biological evaluation of novel inhibitors against cyanobacterial pyruvate dehydrogenase multienzyme complex E1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 19 | 5.96 | 6.13 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4573921 | — | — | 1 | 6.13 |
| CHEMBL4536626 | — | — | 1 | 6.11 |
| CHEMBL4528072 | — | — | 1 | 6.07 |
| CHEMBL4446650 | — | — | 1 | 6.05 |
| CHEMBL4551831 | — | — | 1 | 6.02 |
| CHEMBL4468855 | — | — | 1 | 6.00 |
| CHEMBL4439522 | — | — | 1 | 5.97 |
| CHEMBL4450631 | — | — | 1 | 5.96 |
| CHEMBL4467832 | — | — | 1 | 5.93 |
| CHEMBL4455708 | — | — | 1 | 5.92 |
| CHEMBL4440722 | — | — | 1 | 5.91 |
| CHEMBL4451777 | — | — | 1 | 5.89 |
| CHEMBL4448597 | — | — | 1 | 5.88 |
| CHEMBL4440566 | — | — | 1 | 5.84 |
| CHEMBL604 | CUPRIC SULFATE | 4.0 | 1 | 5.75 |
| CHEMBL1945267 | — | — | 1 | - |
| CHEMBL4462729 | — | — | 1 | - |
| CHEMBL1929455 | — | — | 1 | - |
| CHEMBL1929457 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4573921 | — | EC50 | = | 740.0 | nM | 6.13 |
| CHEMBL4536626 | — | EC50 | = | 780.0 | nM | 6.11 |
| CHEMBL4528072 | — | EC50 | = | 850.0 | nM | 6.07 |
| CHEMBL4446650 | — | EC50 | = | 900.0 | nM | 6.05 |
| CHEMBL4551831 | — | EC50 | = | 950.0 | nM | 6.02 |
| CHEMBL4468855 | — | EC50 | = | 990.0 | nM | 6.00 |
| CHEMBL4439522 | — | EC50 | = | 1060.0 | nM | 5.97 |
| CHEMBL4450631 | — | EC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL4467832 | — | EC50 | = | 1170.0 | nM | 5.93 |
| CHEMBL4455708 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL4440722 | — | EC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL4451777 | — | EC50 | = | 1290.0 | nM | 5.89 |
| CHEMBL4448597 | — | EC50 | = | 1330.0 | nM | 5.88 |
| CHEMBL4440566 | — | EC50 | = | 1430.0 | nM | 5.84 |
| CHEMBL604 | CUPRIC SULFATE | EC50 | = | 1770.0 | nM | 5.75 |
| CHEMBL1945267 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4462729 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1929455 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1929457 | — | EC50 | > | 100000.0 | nM | - |