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Assay Detail

CHEMBL4392268

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Binding
Inhibition of CD73 in human MDA-MB-231 cell membranes using [2,8-3H]AMP as substrate measured after 25 mins by scintillation counting method
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type MDA-MB-231
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

5'-nucleotidase (CHEMBL5957)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structure-Activity Relationship of Purine and Pyrimidine Nucleotides as Ecto-5'-Nucleotidase (CD73) Inhibitors.
Junker A, Renn C, Dobelmann C, Namasivayam V, Jain S, Losenkova K, Irjala H, Duca S, Balasubramanian R, Chakraborty S, Börgel F, Zimmermann H, Yegutkin GG, Müller CE, Jacobson KA.
J Med Chem (2019) 62 : 3677 -3695
PubMed 30895781 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 6 8.11 8.35

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3606064 1 8.35
CHEMBL4483379 1 8.25
CHEMBL4443094 1 8.20
CHEMBL4443977 1 8.10
CHEMBL4551648 1 8.00
CHEMBL4470616 1 7.78

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3606064 Ki = 4.51 nM 8.35
CHEMBL4483379 Ki = 5.68 nM 8.25
CHEMBL4443094 Ki = 6.29 nM 8.20
CHEMBL4443977 Ki = 7.96 nM 8.10
CHEMBL4551648 Ki = 10.1 nM 8.00
CHEMBL4470616 Ki = 16.6 nM 7.78