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Assay Detail

CHEMBL4393881

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Functional
Antileishmanial activity against promastigote stage of Leishmania infantum MHOM/PT/88/IMT151 as parasite growth inhibition after 48 hrs by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania infantum
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania infantum (CHEMBL612848)
Type ORGANISM
Organism Leishmania infantum

Publication

Evaluation of synthetic substituted 1,2-dioxanes as novel agents against human leishmaniasis.
Ortalli M, Varani S, Rosso C, Quintavalla A, Lombardo M, Trombini C.
Eur J Med Chem (2019) 170 : 126 -140
PubMed 30878827 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.25 5.46

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4593142 1 5.46
CHEMBL190579 1 5.03

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4593142 IC50 = 3510.0 nM 5.46
CHEMBL190579 IC50 = 9350.0 nM 5.03