Assay Detail
Functional
CHEMBL4396237
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Antiproliferative activity against human A549 cells assessed as reduction in cell viability at incubated for 72 hrs by MTT assay
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | A549 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Development of novel human lactate dehydrogenase A inhibitors: High-throughput screening, synthesis, and biological evaluations.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 23 | 5.16 | 6.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4065858 | — | — | 1 | 6.44 |
| CHEMBL1436155 | — | — | 1 | 5.24 |
| CHEMBL1559855 | — | — | 1 | 5.11 |
| CHEMBL1440413 | — | — | 1 | 4.83 |
| CHEMBL1611057 | — | — | 1 | 4.72 |
| CHEMBL4450110 | — | — | 1 | 4.64 |
| CHEMBL4556559 | — | — | 1 | - |
| CHEMBL4577089 | — | — | 1 | - |
| CHEMBL4475383 | — | — | 1 | - |
| CHEMBL4441804 | — | — | 1 | - |
| CHEMBL4476280 | — | — | 1 | - |
| CHEMBL4454634 | — | — | 1 | - |
| CHEMBL4461387 | — | — | 1 | - |
| CHEMBL4515658 | — | — | 1 | - |
| CHEMBL4445248 | — | — | 1 | - |
| CHEMBL4462982 | — | — | 1 | - |
| CHEMBL4583436 | — | — | 1 | - |
| CHEMBL4441824 | — | — | 1 | - |
| CHEMBL1256289 | SODIUM OXAMATE | — | 1 | - |
| CHEMBL1554905 | — | — | 1 | - |
| CHEMBL1888862 | — | — | 1 | - |
| CHEMBL4515017 | — | — | 1 | - |
| CHEMBL1555353 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4065858 | — | IC50 | = | 360.0 | nM | 6.44 |
| CHEMBL1436155 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL1559855 | — | IC50 | = | 7800.0 | nM | 5.11 |
| CHEMBL1440413 | — | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL1611057 | — | IC50 | = | 18900.0 | nM | 4.72 |
| CHEMBL4450110 | — | IC50 | = | 22700.0 | nM | 4.64 |
| CHEMBL4556559 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4577089 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4475383 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4441804 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4476280 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4454634 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4461387 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4515658 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4445248 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4462982 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4583436 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4441824 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1256289 | SODIUM OXAMATE | IC50 | = | 45800000.0 | nM | - |
| CHEMBL1554905 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1888862 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4515017 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1555353 | — | IC50 | > | 50000.0 | nM | - |