Assay Detail
Functional
CHEMBL4397637
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Antiproliferative activity against human CTRPA cells harboring APC A1309 mutant after 72 hrs by Celltiter-Glo assay
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Design and Synthesis of TASIN Analogues Specifically Targeting Colorectal Cancer Cell Lines with Mutant Adenomatous Polyposis Coli (APC).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 23 | 8.61 | 10.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4544901 | — | — | 1 | 10.40 |
| CHEMBL4453433 | — | — | 1 | 9.22 |
| CHEMBL4474102 | — | — | 1 | 9.15 |
| CHEMBL4515879 | — | — | 1 | 9.15 |
| CHEMBL4525195 | — | — | 1 | 9.10 |
| CHEMBL4448361 | — | — | 1 | 9.05 |
| CHEMBL4560611 | — | — | 1 | 9.03 |
| CHEMBL4523058 | — | — | 1 | 8.92 |
| CHEMBL4475554 | — | — | 1 | 8.82 |
| CHEMBL4517283 | — | — | 1 | 8.80 |
| CHEMBL4456428 | — | — | 1 | 8.55 |
| CHEMBL4454239 | — | — | 1 | 8.49 |
| CHEMBL4439001 | — | — | 1 | 8.47 |
| CHEMBL4459807 | — | — | 1 | 8.47 |
| CHEMBL4470755 | — | — | 1 | 8.47 |
| CHEMBL4473186 | — | — | 1 | 8.42 |
| CHEMBL4467851 | — | — | 1 | 8.37 |
| CHEMBL4566608 | — | — | 1 | 8.16 |
| CHEMBL4518689 | — | — | 1 | 8.09 |
| CHEMBL4464611 | — | — | 1 | 8.02 |
| CHEMBL4448984 | — | — | 1 | 7.99 |
| CHEMBL4530619 | — | — | 1 | 7.98 |
| CHEMBL4514756 | — | — | 1 | 6.91 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4544901 | — | IC50 | = | 0.04 | nM | 10.40 |
| CHEMBL4453433 | — | IC50 | = | 0.6 | nM | 9.22 |
| CHEMBL4474102 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL4515879 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL4525195 | — | IC50 | = | 0.8 | nM | 9.10 |
| CHEMBL4448361 | — | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL4560611 | — | IC50 | = | 0.94 | nM | 9.03 |
| CHEMBL4523058 | — | IC50 | = | 1.2 | nM | 8.92 |
| CHEMBL4475554 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL4517283 | — | IC50 | = | 1.6 | nM | 8.80 |
| CHEMBL4456428 | — | IC50 | = | 2.8 | nM | 8.55 |
| CHEMBL4454239 | — | IC50 | = | 3.2 | nM | 8.49 |
| CHEMBL4439001 | — | IC50 | = | 3.4 | nM | 8.47 |
| CHEMBL4459807 | — | IC50 | = | 3.4 | nM | 8.47 |
| CHEMBL4470755 | — | IC50 | = | 3.4 | nM | 8.47 |
| CHEMBL4473186 | — | IC50 | = | 3.8 | nM | 8.42 |
| CHEMBL4467851 | — | IC50 | = | 4.3 | nM | 8.37 |
| CHEMBL4566608 | — | IC50 | = | 6.9 | nM | 8.16 |
| CHEMBL4518689 | — | IC50 | = | 8.2 | nM | 8.09 |
| CHEMBL4464611 | — | IC50 | = | 9.6 | nM | 8.02 |
| CHEMBL4448984 | — | IC50 | = | 10.2 | nM | 7.99 |
| CHEMBL4530619 | — | IC50 | = | 10.5 | nM | 7.98 |
| CHEMBL4514756 | — | IC50 | = | 122.0 | nM | 6.91 |