Assay Detail
Binding
CHEMBL4403352
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Inhibition of CDK7 (unknown origin) after 4 hrs
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent advances in the development of cyclin-dependent kinase 7 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.64 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4465061 | — | — | 1 | 7.70 |
| CHEMBL3603847 | — | — | 1 | 7.57 |
| CHEMBL4474655 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4465061 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL3603847 | — | IC50 | = | 27.0 | nM | 7.57 |
| CHEMBL4474655 | — | IC50 | < | 20.0 | nM | - |